Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Found
1
Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [349-460]' and Ligand = 'BDBM391580'
Target
Bromodomain-containing protein 4 [349-460]
(Homo sapiens (Human))
Incyte
US Patent
Ligand
BDBM391580
(2-isopropyl-N-methyl-8-(6- methyl-7-oxo-6,7-dihydr...)
Copy SMILES
Affinity Data
IC50: <100nM
Assay Description:
BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for BD2. Inhib...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI