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TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP1alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Binding affinity at mouse CCR1More data for this Ligand-Target Pair
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