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Found 3 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 4' and Ligand = 'BDBM50363984'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363984(CHEMBL1949730)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-CPCR4 from CXCR4 receptor in human Jurkat cells after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363984(CHEMBL1949730)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]-SDF-1alpha from CXCR4 receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50363984(CHEMBL1949730)
Affinity DataIC50:  63nMAssay Description:Displacement of [125I]SDF-1alpha from CXCR4 expressed in HEK293 cell membrane after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed