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Found 2 Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM150102'
TargetCREB-binding protein(Homo sapiens (Human))
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM150102(US8975417, 170)
Affinity DataIC50:  630nMAssay Description:Inhibition of His-tagged CREBP (unknown origin) using acetyl-histone H4 as substrate after 35 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM150102(US8975417, 170)
Affinity DataIC50:  630nMpH: 7.5 T: 2°CAssay Description:In order to assess bromodomain selectivity, we set up a binding assay using the bromodomain encoded by the CREBBP gene. Compounds were tested in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent