Found 5 Enz. Inhib. hit(s) with Target = 'Calcium/calmodulin-dependent protein kinase type II subunit gamma' and Ligand = 'BDBM2579'
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 0.387nMAssay Description:Inhibition of human CAMK2G using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 0.656nMAssay Description:Inhibition of human CAMK2G using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 0.5nMAssay Description:Average Binding Constant for CAMK2G; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair