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Found 2 Enz. Inhib. hit(s) with Target = 'Calpain-1 catalytic subunit' and Ligand = 'BDBM50265975'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50265975((S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-4-(2,...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human erythrocytes mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50265975((S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-4-(2,...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed