TargetCannabinoid receptor 1/2(Rattus norvegicus (Rat))
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rattus norvegicus (Rat))
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.56nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rattus norvegicus (Rat))
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair