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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50072768'
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072768((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor of rat cerebellar membranes by liquid scintillation counting in presence of serine protease inhibitor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072768((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...)
Affinity DataKi:  173nMAssay Description:Tested for binding affinity to Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072768((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...)
Affinity DataKi:  309nMAssay Description:Binding affinity towards cannabinoid receptor 1 from rat forebrain membranes in the presence of phenylmethanesulfonylfluoride (PMSF) using 0.8 nM [3H...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072768((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((...)
Affinity DataKi:  589nMAssay Description:Binding affinity towards cannabinoid receptor 1 from rat forebrain membranes in the absence of phenylmethanesulfonylfluoride (PMSF) using 0.8 nM [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed