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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50078769'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed