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Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50257659'
TargetCannabinoid receptor 1(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as induction of Ca2+ flux after 10 mins by Fluor-4 AM dye based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  34nMAssay Description:Agonist activity at rat CB1 receptor expressed in mouse AtT20 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  34nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human CB1 receptor expressed in AtT-20 cells measured every 2 secs for 2 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human CB1 receptor expressed in AtT-20 cells measured every 2 secs for 2 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed