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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50513123'
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513123(CHEMBL4576877)
Affinity DataEC50:  17nMAssay Description:Positive allosteric modulation of human Gi/Go-coupled CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced inhibition of for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513123(CHEMBL4576877)
Affinity DataEC50:  828nMAssay Description:Agonist activity at human CB1 receptor expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 30 mins by PathHunt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513123(CHEMBL4576877)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human Gi/Go-coupled CB1 receptor expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513123(CHEMBL4576877)
Affinity DataEC50:  363nMAssay Description:Positive allosteric modulation of human CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced beta-arrestin recruitment prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed