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Report error Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50257659'
TargetCannabinoid receptor 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as induction of Ca2+ flux after 10 mins by Fluor-4 AM dye based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  29nMAssay Description:Antagonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of CP55940-induced Ca2+ flux preincubated for 10 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  29nMAssay Description:Agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human CB2 receptor expressed in AtT-20 cells measured every 2 secs for 2 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50257659(CHEMBL4104511)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human CB2 receptor expressed in AtT-20 cells measured every 2 secs for 2 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed