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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50543738'
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50543738(CHEMBL4644215)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in HEK cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50543738(CHEMBL4644215)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed