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Found 22 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50236959'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]spiperone from human Dopamine D2S receptor expressed in CHO cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]spiperone from human Dopamine D2S receptor expressed in CHO cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]spiperone from human Dopamine D2L receptor expressed in CHO cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]spiperone from human Dopamine D2L receptor expressed in CHO cell membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  6.20nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.40nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.40nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.40nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  275nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human Dopamine D2S receptor expressed in HEK293T cell membranes coexpressing Galphai2 incubated for 30 mins measured after 75 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged Galphai2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged Galphai2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged GalphaoA ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged GalphaoA ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged GalphaoB ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  5.70nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.70nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  2nMAssay Description:Agonist activity at N-terminal flag-tagged D2S receptor (unknown origin) expressed in HEK293 cells coexpressing renilla luciferase 2-tagged GalphaoB ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.40nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50236959(CHEMBL4060461)
Affinity DataEC50:  3.70nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed