Affinity DataKi: 33nMAssay Description:Binding affinity tested against D4.2 receptor in Chinese hamster ovary cell line (CHO cells) using [3H]spiperone as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataEC50: 30.6nMAssay Description:In vitro EC50 tested on HEK293 cells co-transfected with human Dopamine receptor D4.4 using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10.1nMAssay Description:Effective concentration against human Dopamine receptor D4More data for this Ligand-Target Pair