Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'DNA topoisomerase 2-alpha' and Ligand = 'BDBM50242374'
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50242374(CHEMBL505529 | topostatin)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition human placenta topoisomerase 2 assessed as conversion of catenated kinetoplast DNA to minicircle monomerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50242374(CHEMBL505529 | topostatin)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition human placenta topoisomerase 2 assessed as conversion of supercoiled pBR322 DNA to relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed