Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'DNA-(apurinic or apyrimidinic site) endonuclease' and Ligand = 'BDBM222128'
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM222128(7-Chloro-2-(2-fluorophenyl)-4H-3,1-benzoxazin-4-on...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of nuclease activity of APE1 in human glioblastoma cells assessed as reduction in AP site DNA cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed