Found 1 Enz. Inhib. hit(s) with Target = 'DNA-(apurinic or apyrimidinic site) endonuclease' and Ligand = 'BDBM50453749'
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Russian Academy of Sciences
Curated by ChEMBL
Russian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of redox activity of full length N-terminal hexa-His SUMO-fused human APE1 using HEX-labeled THF oligonucleotide as substrate preincubated...More data for this Ligand-Target Pair