Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in rat brain membrane after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to delta-opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]-DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity towards delta-opioid receptor by displacement of [3H]-DADL in rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]diprenorphine from human cloned delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Concentration required to inhibit the binding of the non-selective opioid antagonist, [3H]diprenorphine, to cloned human delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]diprenorphine from human cloned delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:In vitro binding affinity to human Opioid receptor delta 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]naltrindole from human delta-opioid receptor expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Inhibition of [3H]-naltrindole binding to human Opioid receptor delta 1 in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by micro beta2 scintillation c...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H]-diprenorphine from human DOR expressed in CHO cell membranes incubated for 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H]naltrindole from human opioid delta receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor expressed in CHO cell membranes incubated for 1 hr by competition radioligand bin...More data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes measured by competitive radioligand receptor binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Displacement of [3H]-deltorphine from human delta opioid receptor expressed in CHO-K1 cells by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]diprenorphine human delta opioid receptor expressed in CHO cell membranes after 1 hr by micro beta2 scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]Naltrindole form human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataKi: 1.52E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of [3H]DPDPE binding to guinea pig brain membrane Opioid receptor delta 1 at 1.0 nMMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of Opioid receptor delta 1 by displacing 1 nM [3H]DPDPE in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Antagonist activity at human DOR expressed in CHO cell membranes assessed as reduction in SNC80-induced response incubated for 1 hr by [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Antagonist activity at human delta opioid receptor expressed in CHO cell membranes assessed as reduction in SNC80-induced [35S]GTPgammaS binding incu...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Binding affinity against delta-opiate receptor (human) using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Antagonist activity at human delta opioid receptor expressed in CHO cell membranes assessed as reduction in SNC80-induced [35S]GTPgammaS binding prei...More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair