Affinity DataKi: 30nMAssay Description:Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]diprenorphine from human recombinant mu opioid receptor expressed in HEK cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Displacement of [3H]diprenorphine from human opioid delta receptor expressed in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Science and Technology
Curated by ChEMBL
University of Science and Technology
Curated by ChEMBL
Affinity DataKi: >300nMAssay Description:Displacement of [3H]DADLE from delta-opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Science and Technology
Curated by ChEMBL
University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 301nMAssay Description:Binding affinity of compound for opioid receptor delta 1 was determined using [3H]DADLE as radioligand from rat brain tissueMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Science and Technology
Curated by ChEMBL
University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 301nMAssay Description:Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain tissueMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human recombinant delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
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