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Found 1 Enz. Inhib. hit(s) with Target = 'Dimer of Gag-Pol polyprotein [491-589,Q496K]' and Ligand = 'BDBM17827'
TargetDimer of Gag-Pol polyprotein [491-589,Q496K](Human immunodeficiency virus type 1)
University of Massachusetts Medical School

LigandPNGBDBM17827((2S)-2-acetamido-N-[(2S,4S,5S)-4-hydroxy-5-{[(5R)-...)
Affinity DataKi:  131nM ΔG°:  -39.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease inhibitor activities were determined by the fluorescence resonance energy transfer (FRET) method. The energy transfer donor (EDANS) an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed