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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM29609'
TargetEstrogen receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM29609(4-alpha-Cumylphenol | 4-cumylphenol | US9688816, B)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at human Gal4-fused ERalpha expressed in HEK293 cells assessed as inhibition of E2-induced transcriptional activation after 24 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM29609(4-alpha-Cumylphenol | 4-cumylphenol | US9688816, B)
Affinity DataIC50:  1.40E+5nMAssay Description:Competitive binding assays were performed by incubating rhER alpha (α) and beta 1 (β1) receptors with 10 nM [3H]estradiol (the radio ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEstrogen receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM29609(4-alpha-Cumylphenol | 4-cumylphenol | US9688816, B)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at human Gal4-fused ERalpha expressed in HEK293 cells assessed as transcriptional activation after 24 hrs by luciferase/beta-galacto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed