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Found 5 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 35' and Ligand = 'BDBM50259843'
TargetG-protein coupled receptor 35(Homo sapiens (Human))TBA
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataKi:  352nMAssay Description:Competitive binding affinity to Nluc-fused human GPR35 expressed in CHO-K1 cells assessed as inhibition constant using furimazine as substrate incuba...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))TBA
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataIC50:  56nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))TBA
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataEC50:  150nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))TBA
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataEC50:  3.63E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 35(Homo sapiens (Human))TBA
LigandPNGBDBM50259843(CHEMBL4081238)
Affinity DataEC50:  150nMAssay Description:Agonist activity at GPR35 in human HT-29 cells assessed as induction of cell desensitization to 1 uM zaprinast preincubated for 1 hr followed by zapr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed