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Found 1 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 4' and Ligand = 'BDBM50175290'
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175290(CHEMBL3810385)
Affinity DataIC50:  67nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed