Found 2 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-6' and Ligand = 'BDBM50273002'
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University
Curated by ChEMBL
Johannes Gutenberg University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University
Curated by ChEMBL
Johannes Gutenberg University
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at rat recombinant GABAAalpha6beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair