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Found 4 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50006875'
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006875(CHEMBL263969 | N-{(S)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  1.70nMAssay Description:Evaluated for inhibition of cholecystokinin type B receptor by displacing [125I]-Bolton hunter CCK-8 radioligand in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006875(CHEMBL263969 | N-{(S)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of [3H]-propionyl-CCK-8 binding to mouse cerebral cortex membrane cholecystokinin-B (CCK-B) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006875(CHEMBL263969 | N-{(S)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006875(CHEMBL263969 | N-{(S)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  43nMAssay Description:Inhibition of [125I]-CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails Article