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Found 1 Enz. Inhib. hit(s) with Target = 'Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM14452'
LigandPNGBDBM14452(4-[(5-{[5-(naphthalen-1-yl)-1H-indol-1-yl]methyl}-...)
Affinity DataIC50:  270nMAssay Description:The in vitro activity of compounds inhibiting GGTase-1 was determined by measuring the transfer of [3H]-geranylgeranylpyrophosphate to substrate Ha-R...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed