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Found 2 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50120281'
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50120281(CHEMBL3616584)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]glucagon from human glucagon receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50120281(CHEMBL3616584)
Affinity DataIC50:  5nMAssay Description:Antagonist activity against human glucagon receptor expressed in CHO cells assessed as reduction in glucagon-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed