Found 7 Enz. Inhib. hit(s) with Target = 'Glucagon-like peptide 1 receptor' and Ligand = 'BDBM50121400' 
Affinity DataIC50: 0.130nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
Affinity DataKon: 0.123M-1s-1Assay Description:Binding affinity to GLP1R (unknown origin) assessed as dissociation rate constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0190nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
Affinity DataKd: 441nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.00700nMAssay Description:Agonist activity at human GLP1 receptor expressed in BHK cells after 3 hrs by CRE firefly luciferase reporter gene assay in absence of human serum al...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0190nMAssay Description:Activation of GLP1R (unknown origin) CRE-bla expressed in CHO-K1 cells assessed as receptor potency incubated for 1 hrs by time resolved fluorescence...More data for this Ligand-Target Pair
