Report error Found 4 Enz. Inhib. hit(s) with Target = 'Glutamate receptor 1' and Ligand = 'BDBM50252922'
TargetGlutamate receptor 1(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of (R,S)-[5-methyl-3H]AMPA from rat recombinant flop iGluR1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Human)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 374nMAssay Description:Antagonist activity at human flip iGluR1 expressed in CHO-K1 cells by whole cell patch-clamp methodMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 7.20E+3nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR1 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electro...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Human)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at cyclothiazide-desensitized human flip iGluR1 expressed in CHO-K1 cells by whole cell patch-clamp methodMore data for this Ligand-Target Pair