Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 1' and Ligand = 'BDBM50137149'
TargetGlutamate receptor ionotropic, kainate 1(Human)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137149(4-Chloro-2-[3-(3-trifluoromethyl-phenyl)-ureido]-b...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at human homomeric GluR5 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Human)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137149(4-Chloro-2-[3-(3-trifluoromethyl-phenyl)-ureido]-b...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed