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Found
1
Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial' and Ligand = 'BDBM416684'
Target
Glutaminase kidney isoform, mitochondrial
(Homo sapiens (Human))
Astrazeneca
US Patent
Ligand
BDBM416684
((2S)-2-[4-Fluoro-3-(trifluoromethoxy)phenyl]-2-met...)
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Affinity Data
IC50: 69.3nM
Assay Description:
A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...
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Target Info
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Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
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Ligand Info
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US Patent
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