Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM8579'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Tsukuba Research Laboratories

LigandPNGBDBM8579(4-Acylamino-6-arylfuro[2,3-d]pyrimidine 24 | N-[6-...)
Affinity DataIC50:  5nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-32P] ATP. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Tsukuba Research Laboratories

LigandPNGBDBM8579(4-Acylamino-6-arylfuro[2,3-d]pyrimidine 24 | N-[6-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Tsukuba Research Laboratories

LigandPNGBDBM8579(4-Acylamino-6-arylfuro[2,3-d]pyrimidine 24 | N-[6-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human GSK3beta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Tsukuba Research Laboratories

LigandPNGBDBM8579(4-Acylamino-6-arylfuro[2,3-d]pyrimidine 24 | N-[6-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed