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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2 [Y641H]' and Ligand = 'BDBM50009672'
Target
Histone-lysine N-methyltransferase EZH2 [Y641H]
(Homo sapiens (Human))
Epizyme
US Patent
Ligand
BDBM50009672
(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
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Affinity Data
IC50: 263nM
pH: 7.6
Assay Description:
S-Adenosyl-L-homocysteine (SAH) was serially diluted 3 fold in DMSO for 10 points and 1 μL was plated in a 384 well microtiter plate. Positive c...
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