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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50138780'
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50138780(CHEMBL261992 | cyclo[Ala3]Dyn A-(1-11)NH2)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards Opioid receptor kappa 1 expressed in CHO cells was determined by using [3H]-diprenorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50138780(CHEMBL261992 | cyclo[Ala3]Dyn A-(1-11)NH2)
Affinity DataEC50:  0.650nMAssay Description:Inhibition of forskolin-stimulated adenylyl cyclase activity by compound in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed