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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50340646'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50340646(CHEMBL4159127)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in HEK293 cell membranes after 2 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50340646(CHEMBL4159127)
Affinity DataIC50:  0.220nMAssay Description:Agonist activity at human kappa opioid receptor expressed in HEK293 assessed as inhibition forskolin-induced cAMP accumulation after 15 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed