Affinity DataKi: 46nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea-pig brain membranes incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.03E+3nMAssay Description:Agonist activity at human KOR expressed in CHO cell membranes incubated for 60 mins scintillation counting assayMore data for this Ligand-Target Pair