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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 5A/5B' and Ligand = 'BDBM264012'
Target
Lysine-specific demethylase 5A/5B
(Homo sapiens (Human))
Celgene
Curated by
ChEMBL
Ligand
BDBM264012
(2-[5-[(4-chloro-2- methoxyphenyl)methoxy]pyrazol- ...)
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Affinity Data
EC50: 110nM
Assay Description:
Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassay
More data for this Ligand-Target Pair
Target Info
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antibodypedia
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Ligand Info
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