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Found 4 Enz. Inhib. hit(s) with Target = 'Lysine-specific histone demethylase 1A' and Ligand = 'BDBM50548033'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548033(CHEMBL4743670)
Affinity DataIC50:  29nMAssay Description:Inhibition of human recombinant LSD1 using ARTK(diMe)QTARKSTGGKAPRKQLA as substrate incubated for 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548033(CHEMBL4743670)
Affinity DataIC50:  29nMAssay Description:Inhibition of LSD1 (unknown origin) incubated for 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548033(CHEMBL4743670)
Affinity DataIC50:  29nMAssay Description:Inhibition of KDM1A (unknown origin) incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548033(CHEMBL4743670)
Affinity DataIC50:  29nMAssay Description:Inhibition of human LSD1 expressed in Escherichia coli BL21 (DE3) cells using (ARTK(diMe)QTARKSTGGKAPRKQLA peptide as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed