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Report error Found 2 Enz. Inhib. hit(s) with Target = 'MAP kinase-interacting serine/threonine-protein kinase 2' and Ligand = 'BDBM136193'
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM136193(US8853193, 23-2)
Affinity DataIC50:  6nMpH: 7.4 T: 30°CAssay Description:Inhibition of kinase activity of Mnk1 and Mnk2a was assessed with the same assay system, using pre-activated GST-Mnk1 or GST-Mnk2a, respectively. The...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM136193(US8853193, 23-2)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of His-tagged Mnk2 (unknown origin) using eIF4E-derived (D 202 TATKSGSTTKNR 214) peptide as substrate incubated for 90 mins by IMAP TR-FRE...More data for this Ligand-Target Pair
In DepthDetails PubMed