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Found 20 Enz. Inhib. hit(s) with Target = 'Maltase-glucoamylase' and Ligand = 'BDBM23406'
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataKi:  440nMAssay Description:Non-competitive inhibition of alpha glucosidase (unknown origin) assessed as inhibition constant using pNPG as substrate by by Dixon plot analysisMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  172nMAssay Description:Inhibition of alpha glucosidase (unknown origin) using p-nitrophenyl glucopyranoside as substrate by UV Vis- spectrophotometer analysisMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  900nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of human intestinal maltase using maltose as substrate incubated for 30 mins and immediately heated for 2 mins by glucose oxidase methodMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate incubated for 30 mins by absorbance assayMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  2.61E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  3.45E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  3.96E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 3...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by spectrophotometri...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  4.07E+4nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using pNPG as substrate preincubated with enzyme for 15 mins followed by substrate addition and meas...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  2.01E+5nMAssay Description:Inhibition of Alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  2.59E+5nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  4.52E+5nMAssay Description:Inhibition of alpha glucosidase (unknown origin)More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  5.76E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  5.84E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-glycoside as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  7.50E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl glucopyranoside as substrate preincubated for 10 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  7.64E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) by HPLC analysisMore data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  9.06E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin)More data for this Ligand-Target Pair
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  1.52E+6nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate by spectrophotometric assayMore data for this Ligand-Target Pair