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Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50183974'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50183974((E)-6-chloro-4-(1-cinnamylpiperidin-4-ylamino)-1-m...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50183974((E)-6-chloro-4-(1-cinnamylpiperidin-4-ylamino)-1-m...)
Affinity DataIC50:  88nMAssay Description:Inhibition of MCH-mediated calcium release in whole IMR32 cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed