Report error Found 5 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50134955'
Affinity DataKi: 0.220nMAssay Description:Binding affinity against Melanocortin 4 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human MC4R transfected in HEK293 cells co-transfected with GScAMP22F assessed as decrease in alpha-MSH induced cAMP level in p...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human MC4R transfected in HEK293 cells co-transfected with GScAMP22F assessed as decrease in alpha-MSH induced cAMP level in p...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Intracellular cAMP accumulation in Melanocortin 4 receptor functional assay.More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human MC4R transfected in HEK293 cells assessed as cAMP accumulation by competitive binding assayMore data for this Ligand-Target Pair