Report error Found 16 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1C' and Ligand = 'BDBM9019'
Affinity DataKi: 0.176nMAssay Description:Effect of compound on Melatonin receptor in chicken brain in the presence of MnCl2More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor was determined using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.676nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Effect of compound on Melatonin receptor in chicken brain in the presence of GTP-gamma-SMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1C(African clawed frog)
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
TargetMelatonin receptor type 1C(African clawed frog)
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
TargetMelatonin receptor type 1C(African clawed frog)
King'S College London
Curated by PDSP Ki Database
King'S College London
Curated by PDSP Ki Database
Affinity DataEC50: 0.0794nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair