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Report error Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1/3' and Ligand = 'BDBM50456353'
TargetMitogen-activated protein kinase 1/3(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50456353(CHEMBL4210682 | US11001575, Example 2)
Affinity DataIC50:  630nMAssay Description:Inhibition of ERK1/2 in human A375 cells harboring BRAF V600E mutant assessed as suppression of RSK phosphorylation after 4 hrs by MSD assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB