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Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 2' and Ligand = 'BDBM50505542'
TargetMitogen-activated protein kinase kinase kinase 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50505542(CHEMBL4576489)
Affinity DataKd:  53nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged MAP3K2 (unknown origin) (337 to 620 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed