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Found 7 Enz. Inhib. hit(s) with Target = 'Monoglyceride lipase' and Ligand = 'BDBM60419'
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  140nMAssay Description:Inhibition of MAGL in rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat cerebellar membranes MAGL-like activity preincubated for 30 mins followed by 2-AG substrate addition after 90 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  140nMAssay Description:Inhibition of MAGL from Wistar rat brain membranes using 2-AG as substrate after 90 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of human cerebellar membranes MAGL-like activity preincubated for 30 mins followed by 2-AG substrate addition after 90 mins by HPLC analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human MAGL expressed in Escherichia coli using 6-methoxy-4-methylcoumarin ester as substrate after 3 hrs by mass spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed