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Report error Found 1 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM364545'
TargetMu-type opioid receptor(Human)
Purdue Pharma

US Patent
LigandPNGBDBM364545((4bR,6S,8aS,9R)-11-(cyclopropylmethyl)-3- methoxy-...)
Affinity DataKi:  773nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg mem...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent