Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human MOR expressed in CHO cell membranes incubated for 60 mins scintillation counting assayMore data for this Ligand-Target Pair