Found 8 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50263887'
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]NMS from rat muscarinic M1 receptor expressed in CHO cells after 3 hrsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Partial agonist activity at rat muscarinic M1 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
Affinity DataEC50: 6.5nMAssay Description:Agonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 289nMAssay Description:Agonist activity at muscarinic M1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 289nMAssay Description:Agonist activity at muscarinic M1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 255nMAssay Description:Partial agonist activity at human muscarinic M1 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Partial agonist activity at rat muscarinic M1 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
Affinity DataEC50: 255nMAssay Description:Partial agonist activity at human muscarinic M1 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair